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Number of items: 30.

2021

Milne, Kirsty and Sun, Jianhui and Zaal, Esther A. and Mowat, Jenna and Celie, Patrick H.N. and Fish, Alexander and Berkers, Celia R. and Forlani, Giuseppe and Loayza-Puch, Fabricio and Jamieson, Craig and Agami, Reuven (2019) A fragment-like approach to PYCR1 inhibition. Bioorganic and Medicinal Chemistry Letters, 29 (18). pp. 2626-2631. ISSN 0960-894X

McGarry, David H. and Cooper, Ian R. and Walker, Rolf and Warrilow, Catherine E. and Pichowicz, Mark and Ratcliffe, Andrew J. and Salisbury, Anne-Marie and Savage, Victoria J. and Moyo, Emmanuel and Maclean, John and Smith, Andrew and Charrier, Cédric and Stokes, Neil R. and Lindsay, David M. and Kerr, William J. (2018) Design, synthesis and antibacterial properties of pyrimido[4,5-b]indol-8-amine inhibitors of DNA gyrase. Bioorganic and Medicinal Chemistry Letters, 28 (17). pp. 2998-3003. ISSN 0960-894X

Cooper, Ian R. and McCarroll, Andrew J. and McGarry, David and Kirkham, James and Pichowicz, Mark and Walker, Rolf and Warrilow, Catherine and Salisbury, Anne-Marie and Savage, Victoria J. and Moyo, Emmanuel and Forward, Henry and Cheung, Jonathan and Metzger, Richard and Gault, Zoe and Nelson, Gary and Hughes, Diarmaid and Cao, Sha and Maclean, John and Charrier, Cédric and Craighead, Mark and Best, Stuart and Stokes, Neil R. and Ratcliffe, Andrew J. (2016) Discovery and structure-activity relationships of a novel isothiazolone class of bacterial type II topoisomerase inhibitors. Bioorganic and Medicinal Chemistry Letters, 26 (17). pp. 4179-83. ISSN 0960-894X

Cheng, Gang and Muench, Stephen P and Zhou, Ying and Afanador, Gustavo A and Mui, Ernest J and Fomovska, Alina and Lai, Bo Shiun and Prigge, Sean T and Woods, Stuart and Roberts, Craig W and Hickman, Mark R and Lee, Patty J and Leed, Susan E and Auschwitz, Jennifer M and Rice, David W and McLeod, Rima (2013) Design, synthesis, and biological activity of diaryl ether inhibitors of Toxoplasma gondii enoyl reductase. Bioorganic and Medicinal Chemistry Letters, 23 (7). pp. 2035-2043. ISSN 0960-894X

Cowley, Phillip M and Baker, James and Buchanan, Kirsteen I and Carlyle, Ian and Clark, John K and Clarkson, Thomas R and Deehan, Maureen and Edwards, Darren and Kiyoi, Yasuko and Martin, Iain and Osbourn, Dawn and Walker, Glenn and Ward, Nick and Wishart, Grant (2011) Pharmacokinetic optimisation of novel indole-2-carboxamide cannabinoid CB1 antagonists. Bioorganic and Medicinal Chemistry Letters, 21 (7). pp. 2034-2039. ISSN 0960-894X

Kiyoi, Takao and Adam, Julia M and Clark, John K and Davies, Keneth and Easson, Anna-Marie and Edwards, Darren and Feilden, Helen and Fields, Ruth and Francis, Stuart and Jeremiah, Fiona and McArthur, Duncan and Morrison, Angus J and Prosser, Alan and Ratcliffe, Paul D and Schulz, Jurgen and Wishart, Grant and Baker, James and Campbell, Robert and Cottney, Jean E and Deehan, Maureen and Epemolu, Ola and Evans, Louise (2011) Discovery of potent and orally bioavailable heterocycle-based cannabinoid CB1 receptor agonists. Bioorganic and Medicinal Chemistry Letters, 21 (6). pp. 1748-1753. ISSN 0960-894X

Jamieson, Craig and Maclean, John K.F. and Brown, Christopher I and Campbell, Robert A and Gillen, Kevin J. and Gillespie, Jonathan and Kazemier, Bert and Kiczun, Michael and LAMONT, YVONNE and Lyons, Amanda J. and Moir, Elizabeth M. and Morrow, John A. and Pantling, John and Rankovic, Zoran and Smith, Lynn (2011) Structure based evolution of a novel series of positive modulators of the AMPA receptor. Bioorganic and Medicinal Chemistry Letters, 21 (2). pp. 805-811. ISSN 0960-894X

Jamieson, Craig and Campbell, Robert A. and Cumming, Iain A. and Gillen, Kevin J. and Gillespie, Jonathan and Kazemier, Bert and Kiczun, Michael and Lamont, Yvonne and Lyons, Amanda J. and Maclean, John K.F. and Martin, Frederic and Moir, Elizabeth M. and Morrow, John A. and Pantling, John and Rankovic, Zoran and Smith, Lynn (2010) A novel series of positive modulators of the AMPA receptor : structure-based lead optimization. Bioorganic and Medicinal Chemistry Letters, 20 (20). pp. 6072-6075. ISSN 0960-894X

Jamieson, Craig and Basten, Stephanie and Campbell, Robert A. and Cumming, Iain A. and Gillen, Kevin J. and Gillespie, Jonathan and Kazemier, Bert and Kiczun, Michael and Lamont, Yvonne and Lyons, Amanda J. and Maclean, John K.F. and Moir, Elizabeth M. and Morrow, John A. and Papakosta, Marianthi and Rankovic, Zoran and Smith, Lynn (2010) A novel series of positive modulators of the AMPA receptor : discovery and structure based hit-to-lead studies. Bioorganic and Medicinal Chemistry Letters, 20 (19). pp. 5753-5756. ISSN 0960-894X

Letourneau, Jeffrey J and Jokiel, Patrick and Olson, John and Riviello, Christopher M and Ho, Koc-Kan and McAleer, Lihong and Yang, Jingchun and Swanson, Robert N and Baker, James and Cowley, Phillip and Edwards, Darren and Ward, Nick and Ohlmeyer, Michael H J and Webb, Maria L (2010) Identification and hit-to-lead optimization of a novel class of CB1 antagonists. Bioorganic and Medicinal Chemistry Letters, 20 (18). pp. 5449-5453. ISSN 0960-894X

Rankovic, Zoran and Cai, Jiaqiang and Fradera, Xavier and Dempster, Maureen and Mistry, Ashvin and Long, Clive and Hamilton, Emma and King, Angela and Boucharens, Sylviane and Jamieson, Craig and Gillespie, Jonathan and Cumming, Iain and Uitdehaag, Joost and van Zeeland, Mario. (2010) Dioxo-triazines as a novel series of cathepsin K inhibitors. Bioorganic and Medicinal Chemistry Letters, 20 (5). pp. 1488-1490. ISSN 0960-894X