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Article

Halloum, Iman and Viljoen, Albertus and Khanna, Varun and Craig, Derek and Bouchier, Christiane and Brosch, Roland and Coxon, Geoffrey and Kremer, Laurent (2017) Resistance to thiacetazone derivatives active against Mycobacterium abscessus involves mutations in the MmpL5 transcriptional repressor MAB_4384. Antimicrobial Agents and Chemotherapy, 61 (4). e02509-16:1-14. e02509-16. ISSN 0066-4804

Kardar, M. N. and Zhang, T. and Coxon, G. D. and Watson, D. G. and Fearnley, J. and Seidel, V. (2014) Characterisation of triterpenes and new phenolic lipids in Cameroonian propolis. Phytochemistry, 106. pp. 156-163. ISSN 0031-9422

Coxon, Geoffrey and Craig, Derek and Corrales, Rosa Milagros and Vialla, Emilie and Gannoun-Zaki, Laila and Kremer, Laurent (2013) Synthesis, antitubercular activity and mechanism of resistance of highly effective thiacetazone analogues. PLOS One, 8 (1). pp. 1-13. e53162. ISSN 1932-6203

Coxon, Geoffrey and Cooper, Christopher B. and Gillespie, Stephen H. and McHugh, Timothy D. (2012) Strategies and challenges involved in the discovery of new chemical entities during early-stage tuberculosis drug discovery. Journal of Infectious Diseases. ISSN 0022-1899

Berretta, Giacomo and Coxon, Geoffrey (2012) Synthesis of cis,cis-diunsaturated α-meromycolic acid by a palladium-catalysed alkyl–alkyl Negishi reaction. Tetrahedron Letters, 53 (2). pp. 214-216. ISSN 0040-4039

Dover, Lynn G. and Coxon, Geoffrey (2011) Currrent status and research strategies in tuberculosis drug development. Journal of Medicinal Chemistry, 54 (18). 6157–6165. ISSN 0022-2623

Coxon, Geoffrey and Gillespie, Stephen H. (2010) TB- Strength in numbers. Microbiology Today, 2010 (Feb). p. 68. ISSN 1464-0570

Al-Balas, Qosay and Anthony, Nahoum G. and Al-Jaidi, Bilal and Alnimr, Amani and Abbott, Grainne and Brown, Alistair K. and Taylor, Rebecca C. and Besra, Gurdyal S. and McHugh, Timothy D. and Gillespie, Stephen H. and Johnston, Blair F. and Mackay, Simon P. and Coxon, Geoffrey D. (2009) Identification of 2-Aminothiazole-4-Carboxylate derivatives active against mycobacterium tuberculosis H37Rv and the beta-ketoacyl-ACP synthase mtFabH. PLoS One, 4 (5). e5617. ISSN 1932-6203

Coxon, Geoffrey D. and Furman, Brian L. and Harvey, Alan L. and McTavish, John and Mooney, Mark H. and Arastoo, Mahmoud and Kennedy, A.R. and Tettey, J.N.A. and Waigh, R.D. (2009) Benzylguanidines and other galegine analogues inducing weight loss in mice. Journal of Medicinal Chemistry, 52 (11). pp. 3457-3463. ISSN 0022-2623

Mooney, M.H. and Fogarty, S. and Stevenson, C. and Gallagher, A.M. and Palit, P. and Hawley, S.A. and Hardie, D.G. and Coxon, Geoffrey and Waigh, Roger and Tate, R. and Harvey, Alan and Furman, Brian (2008) Mechanisms underlying the metabolic actions of galegine that contribute to weight loss in mice. British Journal of Pharmacology, 153 (8). pp. 1669-1677. ISSN 1476-5381

Clark, Rachael L. and Carter, Katharine C. and Mullen, Alexander B. and Coxon, Geoffrey D. and Owusu-Dapaah, George and McFarlane, Emma and Dao Duong Thi, M. and Grant, M.H. and Tettey, J.N.A. and Mackay, Simon P. (2007) Identification of the benzodiazepines as a new class of antileishmanial agent. Bioorganic and Medicinal Chemistry Letters, 17 (3). pp. 624-627. ISSN 0960-894X

Bhowruth, V. and Brown, A.K. and Reynolds, R.C. and Coxon, G.D. and Mackay, S.P. and Minnikin, D.E. and Besra, G.S. (2006) Symmetrical and unsymmetrical analogues of isoxyl; active agents against mycobacterium tuberculosis. Bioorganic and Medicinal Chemistry Letters, 16 (18). pp. 4743-4747. ISSN 0960-894X

Coxon, G.D. and Al Dulayymi, J.R. and Morehouse, C. and Brennan, P.J. and Besra, G.S. and Baird, M.S. and Minnikin, D.E. (2004) Synthesis and properties of methyl 5-(1R,2S)-(2-octadecylcycloprop-1-yl)pentanoate and other ω-19 chiral cyclopropane fatty acids and esters related to mycobacterial mycolic acids. Chemistry and Physics of Lipids, 127 (1). pp. 35-46. ISSN 0009-3084

Coxon, G.D. and Douglas, J.D. and Minnikin, D.E. (2003) Facile synthesis of (Z)-tetracos-5-enoic acid and racemic cis-4-(2-octadecylcyclopropane-1-yl)-butanoic acid. Chemistry and Physics of Lipids, 126 (1). pp. 49-53. ISSN 0009-3084

Coxon, G.D. and Al Dulayymi, J.R. and Baird, M.S. and Knobl, S. and Roberts, E. and Minnikin, D.E. (2003) The synthesis of (11R,12S)-lactobacillic acid and its enantiomer. Tetrahedron: Asymmetry, 14 (9). pp. 1211-1222. ISSN 1362-511X

Book Section

Coxon, Geoffrey; (2011) b-antiTB drugs. In: Pharmaceutical and Medical Chemistry. Elsevier. ISBN 9780443072321

Conference or Workshop Item

Coxon, Geoffrey (2012) Strategies and challenges involved in the discovry of new chemical entities during early-stage tuberculosis drug discovery. In: Tuberculosis: Local and global, 2012-03-23.

Coxon, Geoffrey (2011) Discovery and development of new TB drugs. In: All Parliamentary Group on Global Tuberculosis, 2011-06-06.

Coxon, Geoffrey (2009) Medicinal chemistry strategies in combating antibiotic resistance. In: Antibiotic Resistance: From genes to global prevalence, 2009-12-01.

Coxon, Geoffrey (2009) The identification of 2-aminothiazole-4-carboxylates active against Mycobacterium tuberculosis. In: Gordon Research conference on TB Drug Development, 2011-03-31.

Report

Coxon, Geoffrey (2011) The UK's response to global tuberculosis. APPG on Global Tuberculosis.

Other

Coxon, Geoffrey (2012) Written Evidence from TBD-UK, Dr Geoff Coxon. UK Parliament.