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2023
Henry, Martyn C. and Riley, Christopher M. and Hunter, Irene and Elwood, Jessica. M. L. and Lopez-Fernandez, J. Daniel and Minty, Laura and Coe, Diane M. and McEwan, Iain J. and Jamieson, Craig (2023) Synthesis and evaluation of small molecule inhibitors of the androgen receptor N-terminal domain. ACS Medicinal Chemistry Letters, 14 (12). pp. 1800-1806. ISSN 1948-5875
2021
Clegg, Michael A. and Theodoulou, Natalie H. and Bamborough, Paul and Chung, Chun-wa and Craggs, Peter D. and Demont, Emmanuel H. and Gordon, Laurie J. and Liwicki, Gemma M. and Phillipou, Alex and Tomkinson, Nicholas C. O. and Prinjha, Rab K. and Humphreys, Philip G. (2021) Optimization of naphthyridones into selective TATA-binding protein associated factor 1 (TAF1) bromodomain inhibitors. ACS Medicinal Chemistry Letters, 12 (8). pp. 1308-1317. ISSN 1948-5875
2020
Spencer, Jonathan A. and Baldwin, Ian R. and Barton, Nick and Chung, Chun-Wa and Convery, Máire A. and Edwards, Christopher D. and Jamieson, Craig and Mallett, David N. and Rowedder, James E. and Rowland, Paul and Thomas, Daniel A. and Hardy, Charlotte J. (2020) Design and development of a macrocyclic series targeting phosphoinositide 3-kinase δ. ACS Medicinal Chemistry Letters, 11 (7). pp. 1386-1391. ISSN 1948-5875
2018
Ahonen, Tiina J. and Savinainen, Juha R. and Yli-Kauhaluoma, Jari and Kalso, Eija and Laitinen, Jarmo T. and Moreira, Vânia M. (2018) Discovery of 12-thiazole abietanes as selective inhibitors of the human metabolic serine hydrolase hABHD16A. ACS Medicinal Chemistry Letters, 9 (12). pp. 1269-1273. ISSN 1948-5875
2016
Measom, Nicholas and Down, Kenneth D. and Hirst, David J. and Jamieson, Craig and Manas, Eric S. and Patel, Vipulkumar K. and Somers, Donald O. (2016) Investigation of a bicyclo[1.1.1]pentane as a phenyl replacement within an LpPLA2 inhibitor. ACS Medicinal Chemistry Letters, 7.
2015
Caldwell, Nicola and Harms, Jonathan E. and Partin, Kathryn M. and Jamieson, Craig (2015) Rational design of a novel AMPA receptor modulator through a hybridization approach. ACS Medicinal Chemistry Letters.