Browse by Author or creator

2025

Ahmed, Ikhlas M. M. and Rofe, Adam and Henry, Martyn C. and West, Eric and Jamieson, Craig and McEwan, Iain J. and Beveridge, Rebecca (2025) Ion mobility mass spectrometry unveils conformational effects of drug lead EPI-001 on the intrinsically disordered N-terminal domain of the Androgen Receptor. Protein Science, 34 (1). e5254. ISSN 1469-896X

2024

Henry, Martyn C. and Minty, Laura and Kwok, Alexander C. W. and Elwood, Jessica M. L. and Foulis, Adam J. and Pettinger, Jonathan and Jamieson, Craig (2024) One-pot oxidative amidation of aldehydes via the generation of nitrile imine intermediates. Journal of Organic Chemistry, 89 (11). pp. 7913-7926. ISSN 0022-3263

2023

Henry, Martyn C. and Riley, Christopher M. and Hunter, Irene and Elwood, Jessica. M. L. and Lopez-Fernandez, J. Daniel and Minty, Laura and Coe, Diane M. and McEwan, Iain J. and Jamieson, Craig (2023) Synthesis and evaluation of small molecule inhibitors of the androgen receptor N-terminal domain. ACS Medicinal Chemistry Letters, 14 (12). pp. 1800-1806. ISSN 1948-5875

Riley, Christopher M. and Elwood, Jessica M. L. and Henry, Martyn C. and Hunter, Irene and Lopez-Fernandez, J. Daniel and McEwan, Iain J. and Jamieson, Craig (2023) Current and emerging approaches to noncompetitive AR inhibition. Medicinal Research Reviews, 43 (5). pp. 1701-1747. ISSN 0198-6325

Henry, Martyn C. and Anderson, Jack Q. and Jamieson, Craig (2023) Multigram-scale synthesis of a gem-difluoro-substituted 4,5,6,7-tetrahydrobenzo[c]thiophen-4-one heterocycle via oxidative chlorination and radical Smiles rearrangement. Synlett, 34. ISSN 0936-5214

2022

Elwood, Jessica M. L. and Henry, Martyn C. and Lopez-Fernandez, J. Daniel and Mowat, Jenna M. and Boyle, Mhairi and Buist, Benjamin and Livingstone, Keith and Jamieson, Craig (2022) Functionalized tetrazoles as latent active esters in the synthesis of amide bonds. Organic Letters, 24 (51). pp. 9491-9496. ISSN 1523-7060

Boyle, Mhairi and Livingstone, Keith and Henry, Martyn C. and Elwood, Jessica M. L. and Lopez Fernandez, J. Daniel and Jamieson, Craig (2022) Amide bond formation via the rearrangement of nitrile imines derived from N-2-nitrophenyl hydrazonyl bromides. Organic Letters, 24 (1). pp. 334-338. ISSN 1523-7060

2021

Milne, Kirsty and Henry, Martyn C. and Jamieson, Craig (2021) Synthesis of an allylic gem-difluoromethylene building block via radical-mediated difluorocyclopropane ring opening. Tetrahedron Letters, 81. 153344. ISSN 0040-4039