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2024

Hryczanek, Ross P. and Hackett, Andrew S. and Rowland, Paul and Chung, Chun-wa and Convery, Máire A. and Holmes, Duncan S. and Hutchinson, Jonathan P. and Kitchen, Semra and Korczynska, Justyna and Law, Robert P. and Lea, Jonatahn D. and Liddle, John and Lonsdale, Richard and Neu, Margarete and Nickels, Leng and Phillipou, Alex and Rowedder, James E. and Schneck, Jessica L. and Scott-Stevens, Paul and Sheehan, Hester and Tayler, Chloe L. and Temponeras, Ioannis and Tinworth, Christopher P. and Walker, Ann L. and Wojno-Picon, Justyna and Young, Robert J. and Lindsay, David M. and Stratikos, Efstratios (2024) Optimization of potent and selective cyclohexyl acid ERAP1 inhibitors using structure- and property-based drug design. ACS Medicinal Chemistry Letters, 15 (12). 2107–2114. ISSN 1948-5875

2019

Tinworth, Christopher P. and Lithgow, Hannah and Dittus, Lars and Bassi, Zuni I. and Hughes, Sophie E. and Muelbaier, Marcel and Dai, Han and Smith, Ian E. D. and Kerr, William J. and Burley, Glenn A. and Bantscheff, Marcus and Harling, John D. (2019) PROTAC-mediated degradation of Bruton's tyrosine kinase is inhibited by covalent binding. ACS Chemical Biology, 14 (3). pp. 342-347. ISSN 1554-8937