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2023

Aatkar, Arron and Vuorinen, Aini and Longfield, Oliver E. and Gilbert, Katharine and Peltier-Heap, Rachel and Wagner, Craig D. and Zappacosta, Francesca and Rittinger, Katrin and Chung, Chun-wa and House, David and Tomkinson, Nicholas C. O. and Bush, Jacob T. (2023) Efficient ligand discovery using sulfur(VI) fluoride reactive fragments. ACS Chemical Biology. ISSN 1554-8937

Gilbert, Katharine E. and Vuorinen, Aini and Aatkar, Arron and Pogány, Peter and Pettinger, Jonathan and Grant, Emma K. and Kirkpatrick, Joanna M. and Rittinger, Katrin and House, David and Burley, Glenn A. and Bush, Jacob T. (2023) Profiling sulfur(VI) fluorides as reactive functionalities for chemical biology tools and expansion of the ligandable proteome. ACS Chemical Biology, 18 (2). pp. 285-295. ISSN 1554-8937

2021

Fournier, Julie C. L. and Evans, John P. and Zappacosta, Francesca and Thomas, Daniel A. and Patel, Vipulkumar K. and White, Gemma V. and Campos, Sebastien and Tomkinson, Nicholas C. O. (2021) Acetylation of the catalytic lysine inhibits kinase activity in PI3Kδ. ACS Chemical Biology, 16 (9). pp. 1644-1653. ISSN 1554-8937

2019

Tinworth, Christopher P. and Lithgow, Hannah and Dittus, Lars and Bassi, Zuni I. and Hughes, Sophie E. and Muelbaier, Marcel and Dai, Han and Smith, Ian E. D. and Kerr, William J. and Burley, Glenn A. and Bantscheff, Marcus and Harling, John D. (2019) PROTAC-mediated degradation of Bruton's tyrosine kinase is inhibited by covalent binding. ACS Chemical Biology, 14 (3). pp. 342-347. ISSN 1554-8937

2017

Sadler, Joanna C. and Chung, Chun-wa H. and Mosley, Julie E. and Burley, Glenn A. and Humphreys, Luke D. (2017) Structural and functional basis of C-methylation of coumarin scaffolds by NovO. ACS Chemical Biology, 12 (2). pp. 374-379. ISSN 1554-8937